Skip to main content
CSTSetup
Dictionary · Drug

theophylline

A bronchodilator taken by mouth that relaxes and opens the airways, used long term for asthma and COPD.

thee-OFF-ih-lin noun

What it means

A methylxanthine, a drug related to caffeine. It relaxes the smooth muscle of the airways and is used for long-term control of asthma and COPDsee-oh-pee-dee (said as letters)Chronic obstructive pulmonary disease: a long-term lung disease that makes it hard to move air out of the lungs.chronic long-lastingobstructive blockingpulmon/o lung-ary relating toFull entry , though newer inhalers have mostly replaced it. Its safe range is narrow, so blood levels are checked. Too much causes nausea, vomiting, restlessness, a fast heart rate and, at high levels, dangerous heart rhythms and seizures.

For the nurse

Teach the client to limit caffeine (coffee, tea, cola, chocolate), which adds to its effects, and to tell the provider about starting or stopping smoking, which changes drug levels. Many drugs, such as cimetidine and some antibiotics, raise its level. Extended-release forms are swallowed whole.

At a glance

Normal rangeTherapeutic blood level about 10–20 mcg/mL [55–110 µmol/L]; many prescribers aim lower (5–15 mcg/mL).
Drug classbronchodilator (methylxanthine)
Brand namesTheo-24, Elixophyllin
Spanishteofilina
Also writtenTheo-24, Elixophyllin

Related terms

COPD

Chronic obstructive pulmonary disease: a long-term lung disease that makes it hard to move air out of the lungs.

salmeterol

A long-acting inhaled bronchodilator, used twice a day to keep the airways open in asthma and COPD.

cimetidine

An H2 blocker taken by mouth that lowers the amount of acid the stomach makes.

Filed under

Look up another word